TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0570nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0670nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0850nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0850nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.75nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Info
In DepthDetails
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Info
In DepthDetails
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Info
In DepthDetails
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human PNP activityMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human PNP activityMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human PNP activityMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Info
In DepthDetails
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human PNP activityMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 9.5nMAssay Description:Inhibition of human erythrocyte PNP assessed as inhibition of 25 uM 7-methylguanosine phosphorolysis by spectrophotometry in presence of 1 mM inorgan...More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 9.5nMAssay Description:Inhibition of human PNP in presence of 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant PNP using MSEG as substrate preincubated with inhibitor within 10 to 20 mins measured after 5 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Info
In DepthDetails
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human PNP activityMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 20.2nMAssay Description:Inhibition of human PNP in presence of 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 20.2nMAssay Description:Inhibition of human erythrocyte PNP assessed as inhibition of 25 uM 7-methylguanosine phosphorolysis by spectrophotometry in presence of 1 mM inorgan...More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 20.4nMAssay Description:Inhibition of human PNP in presence of 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 20.4nMAssay Description:Inhibition of human erythrocyte PNP assessed as inhibition of 25 uM 7-methylguanosine phosphorolysis by spectrophotometry in presence of 1 mM inorgan...More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human erythrocyte PNP assessed as inhibition of 25 uM 7-methylguanosine phosphorolysis by spectrophotometry in presence of 1 mM inorgan...More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human purine nucleoside phosphorylaseMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 50 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 50 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Compound was evaluated for inhibition of PNP-catalyzed inosine phosphorylation in Cellulomonas spMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Compound was evaluated for inhibition of PNP-catalyzed inosine phosphorylation in Cellulomonas spMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair